Repeat doses of BAY1902607 in healthy males & PoC in chronic cough pts

  • Research type

    Research Study

  • Full title

    Two-part, double-blind, placebo-controlled, randomized, parallel-group study: (Part 1) in healthy male subjects to assess safety and tolerability of ascending repeated oral doses of BAY 1902607 including its effect on the pharmacokinetics of a sub-therapeutic dose of midazolam (MDZ), followed by (Part 2) a two-way crossover administration of four different doses of BAY 1902607 in patients with refractory chronic cough to assess safety, tolerability and efficacy for proof of concept

  • IRAS ID

    242717

  • Contact name

    Tatjana Gust

  • Contact email

    tatjana.gust@bayer.com

  • Sponsor organisation

    Bayer AG

  • Eudract number

    2018-000129-29

  • Duration of Study in the UK

    0 years, 11 months, 31 days

  • Research summary

    This study will investigate the safety and tolerability of ascending repeated oral doses of BAY 1902607 in healthy subjects plus the effect of BAY 1902607 on the pharmacokinetics (PK) of a sub-therapeutic 1 mg dose of midazolam (Part 1). This study will also investigate the safety, tolerability and efficacy of BAY 1902607 in patients with refractory chronic cough (Part 2).

    Part 1 of the study is a randomized, placebo-controlled, double-blind, sequential parallel-group design with repeated doses of BAY 1902607 or placebo administered over 2 weeks. In each dose cohort 12 subjects will be included (9 receiving active, 3 receiving placebo). 4 different ascending doses will be administered in the study. Dosing will start with the lowest dose; escalation to each higher dose of BAY 1902607 will only take place according to specified rules after review of safety, tolerability and PK data from the preceding dose group.

    In each dose group, subjects will also receive a sub-therapeutic dose of midazolam on Day -1 and Day 13 allowing an intraindividual comparison of the drug-drug interaction for subinduction of midazolam.

    Part 2 of the study is two-arm crossover design with repeated doses of BAY 1902607 or placebo administered over two periods (Period A, Period B) of 16 days each, with a 3- to 4-week washout period between the two periods. In Period A, the 4 ascending doses of BAY 1902607 will be given (each dose for 4 days); in Period B, the matching placebo doses will be administered. The patients will be randomized to a treatment sequence of either Period A-Period B or Period B-Period A (crossover principle).

  • REC name

    North West - Greater Manchester Central Research Ethics Committee

  • REC reference

    18/NW/0098

  • Date of REC Opinion

    8 May 2018

  • REC opinion

    Further Information Favourable Opinion