GS-US-401-1787,Open label Study - Long-term Safety of ONO/GS-4059

  • Research type

    Research Study

  • Full title

    An Open-label Study to Assess the Long-term Safety and Efficacy of ONO/GS-4059 in Subjects with Relapsed/Refractory B-cell malignancies.

  • IRAS ID

    184150

  • Contact name

    Martin Dyer

  • Contact email

    mjsd1@le.ac.uk

  • Sponsor organisation

    Gilead Sciences, Inc.

  • Eudract number

    2015-001404-58

  • Clinicaltrials.gov Identifier

    NCT02457559

  • Duration of Study in the UK

    4 years, 0 months, 0 days

  • Research summary

    The purpose of this study is to determine the long-term safety and tolerability of ONO/GS-4059 in subjects in a prior ONO/GS-4059 study and whose disease had not progressed on the parent study.

    ONO/GS-4059, is a small molecule inhibitor of Bruton’s tyrosine kinase (BTK) in the treatment of B-cell malignancies. It was initially evaluated in a Phase 1 single agent dose escalation study, ONO-4059POE001, conducted in the United Kingdom (UK). As of January 2015, this study has enrolled and treated approximately 90 subjects with relapsed CLL, non-GCB DLBCL, MCL, SLL, and other indolent non-Hodgkin’s lymphomas (iNHLs). Tolerability and efficacy were demonstrated in subjects with CLL at doses ranging from 40 to 600 mg once daily with no maximum tolerated dose (MTD) identified. Responses were observed in subjects in the NHL cohort at doses from 40 to 480 mg. Dose limiting toxicities (DLTs) of rash, and non-immune reaction were observed at 600 mg once daily in the NHL cohort.

    Many patients that are currently on treatment with GS-4059 have had no significant adverse events were seen in patients currently on GS-4059 and the efficacy of this drug was shown to be good.

    The study will take place at about 3 centres in the United Kingdom. There will be approximately 32 patients. The study will last approximately 2 years.

  • REC name

    West Midlands - Edgbaston Research Ethics Committee

  • REC reference

    15/WM/0263

  • Date of REC Opinion

    15 Sep 2015

  • REC opinion

    Further Information Favourable Opinion