Evaluating oral BCX9930 in renal disease

  • Research type

    Research Study

  • Full title

    An Open-Label, Safety, Tolerability, and Proof-of-Concept Study of Oral BCX9930 Therapy in Subjects with Complement 3 Glomerulopathy, Immunoglobulin A Nephropathy, or Primary Membranous Nephropathy

  • IRAS ID

    297898

  • Contact name

    Kathryn Hutchinson

  • Contact email

    kathryn.hutchinson@ams-europe.com

  • Sponsor organisation

    BioCryst Pharmaceuticals Inc

  • Eudract number

    2020-005855-19

  • Clinicaltrials.gov Identifier

    NCT05162066

  • Duration of Study in the UK

    2 years, 0 months, 0 days

  • Research summary

    Summary of research
    The study will assess the efficacy and safety of daily oral treatment of BCX9930 in three different renal diseases.
    BCX9930 is a Factor D inhibitor. Factor D is the rate limiting enzyme in the alternative pathway of the complement cascade.
    The study will assess participants with either C3G (Complement 3 Glomerulopathy), or IgA Nephropathy or PMN (Primary Membranous Nephropathy). All three diseases have been associated with alterations in the complement pathway, have limited treatment options and will eventually lead to ESRD.
    The study is open label, and will treat approximately 14 participants in each of the three cohorts. Participants will be treated for 24 weeks, as chronic renal indications typically require long treatment periods to see an improvement in renal function.

    Summary of Results
    In December 2022, BioCryst stopped development of BCX9930 based on changes in the competitive environment. Therefore, this study was prematurely discontinued. A total of 3 subjects were screened and 2 subjects were administered BCX9930.

  • REC name

    East Midlands - Nottingham 2 Research Ethics Committee

  • REC reference

    21/EM/0182

  • Date of REC Opinion

    13 Aug 2021

  • REC opinion

    Further Information Favourable Opinion