A study to assess the safety, tolerability, PK and PD of LAS190792

  • Research type

    Research Study

  • Full title

    A 2-PART, RANDOMISED, PLACEBO-CONTROLLED, SAFETY, TOLERABILITY, PHARMACOKINETIC AND PHARMACODYNAMIC STUDY OF LAS190792 DELIVERED BY INHALATION IN ASTHMATIC AND CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) SUBJECTS.

  • IRAS ID

    132753

  • Contact name

    Tim Mant

  • Contact email

    tim.mant@quintiles.com

  • Sponsor organisation

    Almirall S.A.

  • Eudract number

    2013-001758-93

  • ISRCTN Number

    N/A

  • Clinicaltrials.gov Identifier

    N/A

  • Research summary

    LAS190792 is a new chemical entity possessing long-acting dual-pharmacology activity (muscarinic receptor antagonism and beta2 adrenoceptor agonism (MABA) in a single molecule, which is being developed by Almirall for the treatment of Chronic Obstructive Pulmonary Disease (COPD) and potentially asthma. Blocking of these receptors by other drugs has been shown to be of value in the management of asthma / COPD. The study has two parts; a single ascending dose study in males volunteers with mild persistent asthma and a 5 way crossover (each patient takes a different dose / medication on each of the 5 occasions), single dose study in males and non-childbearing women volunteers with moderate to severe COPD. The purpose of the study is to examine the safety, tolerability, the pharmacodynamics (what the drug does to the body) and pharmacokinetics (the way the body handles absorbs, distributes, breaks down and excretes) various doses of LAS190792 in patients with mild persistent asthma and patients with moderate to severe COPD. This will be the first time LAS190792 has been given to human subjects, and the study has been designed to provide data on which to base future work to establish the safety, the tolerability and the efficacy profile of LAS190792 in treating patients with asthma and COPD.

  • REC name

    West Midlands - Coventry & Warwickshire Research Ethics Committee

  • REC reference

    13/WM/0292

  • Date of REC Opinion

    21 Aug 2013

  • REC opinion

    Further Information Favourable Opinion