A Phase 1 Study to Evaluate ALN-HSD in HV and Adult Patients with NASH

  • Research type

    Research Study

  • Full title

    A Phase 1, Randomized, Double-Blind, Placebo-Controlled, 2-Part Study of the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Single Dose ALN-HSD in Healthy Adult Subjects and Multiple Dose ALN-HSD in Adult Patients with Nonalcoholic Steatohepatitis (NASH)

  • IRAS ID

    286227

  • Contact name

    Jorg Taubel

  • Contact email

    j.taubel@richmondpharmacology.com

  • Sponsor organisation

    Alnylam UK Limited

  • Eudract number

    2020-000847-29

  • Duration of Study in the UK

    0 years, 10 months, 17 days

  • Research summary

    Non-alcoholic fatty liver disease (NAFLD) is the most rapidly growing cause of liver-related mortality and morbidity, affecting 25% of the global adult population [Paik 2020; Younossi 2019a]. The prevalence of non-alcoholic steatohepatitis (NASH) in the United States (US), Europe, and other developed countries is between 1.5% and 6.5%, and it is estimated that 7% to 30% of NAFLD patients progress to NASH [Farrell and Larter 2006; Williams 2011; Younossi 2016]. There are currently no approved pharmacological treatments for NASH, despite the rising burden and increasing NASH prevalence.

    ALN-HSD is a novel synthetic RNA interference (RNAi) therapeutic in development for the treatment of NASH. ALN-HSD contains a small interfering RNA (siRNA) targeting hydroxysteroid 17β dehydrogenase 13 messenger RNA (HSD17β13 mRNA). Based on the mechanism of RNA interference, ALN-HSD is specifically designed to reduce the liver synthesis of HSD17B13 protein. By doing this it is anticipated that ALN-HSD will halt and/or reduce liver injury, fibrosis, and inflammation that occur in NASH.

    This study will be conducted in 2 parts: Part A; a single ascending dose part in healthy adult subjects, and Part B; a multiple dosing part in adult patients with NASH.

  • REC name

    London - London Bridge Research Ethics Committee

  • REC reference

    20/LO/0891

  • Date of REC Opinion

    17 Sep 2020

  • REC opinion

    Further Information Favourable Opinion